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A Case Approach to Perioperative Drug-Drug InteractionsPharmacokinetic Interactions: Core Concepts

A Case Approach to Perioperative Drug-Drug Interactions: Pharmacokinetic Interactions: Core Concepts [This chapter discusses the essential terms and concepts pertaining to how the body processes drugs. This subset of pharmacology is known as pharmacokinetics.] http://www.deepdyve.com/assets/images/DeepDyve-Logo-lg.png

A Case Approach to Perioperative Drug-Drug InteractionsPharmacokinetic Interactions: Core Concepts

Editors: Marcucci, Catherine; Hutchens, Michael P.; Wittwer, Erica D.; Weingarten, Toby N.; Sprung, Juraj; Nicholson, Wayne T.; Lalwani, Kirk; Metro, David G.; Dull, Randal O.; Swide, Christopher E.; Seagull, F. Jacob; Kirsch, Jeffrey R.; Sandson, Neil B.

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References (12)

Publisher
Springer New York
Copyright
© Springer Science+Business Media New York 2015
ISBN
978-1-4614-7494-4
Pages
15 –22
DOI
10.1007/978-1-4614-7495-1_3
Publisher site
See Chapter on Publisher Site

Abstract

[This chapter discusses the essential terms and concepts pertaining to how the body processes drugs. This subset of pharmacology is known as pharmacokinetics.]

Published: May 7, 2013

Keywords: Pharmacokinetics; Pharmacodynamics; Distribution; Metabolism; Excretion; Bioavailability; Hepatic extraction; Morphine; Absorption; Transporters; P-glycoprotein; P-gp; Organic anion-transporting peptide; OATP; Efflux transporter; Grapefruit juice; Fexofenadine CYP3A4; Substrate; Inducer; Inhibitor; Midazolam; Plasma concentration; Peak concentration; Trough; Volume of distribution; Warfarin; Protein binding; Digoxin; Albumin; Free fraction; Unbound fraction; Liver failure; Nephrotic syndrome; Heart failure; Phase I metabolism; Phase II metabolism; Oxidation; Reduction; Hydrolysis; Steroid hormones; Cytochrome; CYP450; Cytochrome; P450; CYP; 3A5; 3A7; 2C9; 2D6; Conjugation; Glucuronidation; Competitive inhibition; CYP3A5; CYP3A7; Clarithromycin; Itraconazole; Ketoconazole; Rifampin; Carbamazepine; St. John’s wort; Carbamazepine; Valproic acid; CYP2C9; Prodrug; CYP2D6; Tamoxifen; Endoxifen; Venlafaxine; Sertraline; Citalopram; Fluoxetine; Paroxetine; Pharmacogenomics; Poor metabolizer; Intermediate metabolizer; Extensive metabolizer; Ultra-rapid metabolizer; Beta-blocker; Metoprolol; Carvedilol; Codeine; Total drug clearance; Famotidine; Glomerular filtration rate; Creatinine clearance; Cockcroft-Gault formula; Modification of Diet in Renal Disease formula; Probenicid; Penicillin; First-order kinetics; Zero-order kinetics; Context-sensitive half-time

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